Development Pipeline

Our Pipeline

Focused innovation with STAT3 as our anchor target, transforming 'undruggable' challenges into breakthrough therapies for fibrosis and oncology.

TTI-101: Our Lead Candidate

An oral small molecule inhibitor selectively targeting the STAT3 SH2 domain

Mechanism of Action

TTI-101 is designed to selectively bind to the SH2 domain of STAT3, blocking pathological signaling that drives disease progression in fibrosis and cancer while maintaining minimal off-target toxicity.

Selective Targeting

Precisely binds to the STAT3 SH2 domain with high specificity, avoiding off-target effects.

Disrupts Pathological Signaling

Prevents STAT3 dimerization and nuclear translocation, blocking transcription of disease-promoting genes.

Demonstrated Efficacy

Shown robust activity in preclinical models of IPF and HCC, with promising early clinical data.

STAT3 Signaling Pathway

The STAT3 pathway plays a crucial role in fibrosis, inflammation, and tumor progression. TTI-101 specifically targets the SH2 domain, blocking the pathological effects while preserving normal cellular function.

Clinical Trials

Our lead candidate TTI-101 is being evaluated in two key clinical trials with near-term catalysts

Phase 2
Enrollment Complete

RENEW-IPF Trial

Evaluating TTI-101 in patients with Idiopathic Pulmonary Fibrosis, a progressive lung disease with high unmet need.

Trial Status:Data Analysis
Patients Enrolled:86
Primary Endpoint:Change in FVC at 24 weeks
Topline Results:Q4 2025
Progress90%
Phase 1b/2
Ongoing

RECLAIM-HCC Trial

Evaluating TTI-101 as monotherapy and in combination with standard-of-care in advanced Hepatocellular Carcinoma.

Trial Status:Patient Recruitment
Patients Target:120
Primary Endpoint:Objective Response Rate
Topline Results:Mid-2026
Progress65%

Pipeline Overview

Our development programs span multiple indications with a focus on fibrosis and oncology

Program
Discovery
Preclinical
Phase 1
Phase 2
Phase 3
TTI-101
Idiopathic Pulmonary Fibrosis
TTI-101
Hepatocellular Carcinoma
NC-201
Systemic Sclerosis
NC-202
NSCLC
Completed
Phase 2 - Ongoing
Phase 1b/2 - Ongoing
IND-Enabling
Lead Optimization
Partner With Us

Partnering Opportunities

We are seeking strategic partnerships to accelerate our pipeline development and expand the therapeutic potential of our proprietary STAT3 platform.

Co-development partnerships

Licensing opportunities

Research collaborations

Strategic investments